Hematology: Coagulation Cascade
Coagulation Cascade
Initial Injury
- Induces:
- Vasoconstriction
- Platelet Adhesion
- Thrombin Release
- Initiates the Intrinsic & Extrinsic Pathways
Intrinsic Pathway
- Initiated By: Exposed Collagen, Pre-Kallikrein, HMW Kininogen
- Pathway:
- Activated Factor XII Activates Factor XI
- Activated Factor XI Activates Factor IX
- Activated Factor IX & VIII Activates Factor X
- Associated Factors: Factor 8, 9, 10, 11 & 12
Extrinsic Pathway
- Initiated By: Tissue Factor (Injured Cells)
- Pathway:
- Activated Factor VII Activates Factor X
- Associated Factors: Factor 7 & 10
Common Pathway
- Initiated By: Intrinsic or Extrinsic Pathways
- Pathway:
- Prothrombin Complex: Activated Factor X, Factor V, Platelet Factor 3 & Prothrombin
- Converts Prothrombin (Factor II) to Thrombin
- Thrombin Converts Fibrinogen (Factor I) to Fibrin
- Prothrombin Complex: Activated Factor X, Factor V, Platelet Factor 3 & Prothrombin
- Thrombin (Factor IIa)
- Converts Fibrinogen to Fibrin
- Also Activates Factors V, VIII & XIII
- Activates Platelets
- Fibrin (Factor Ia)
- Links Platelets to Form a Platelet Plug
- Binds GpIIb/IIIa
- Fibrin Stabilizing Factor (Factor XIII)
- Activated by Thrombin
- Crosslinks Fibrin to Improve Clot Stability
Mediators of Coagulation
Factor Synthesis
- Factor VIII:
- Produced in the Endothelium with vWF
- All Other Factors:
- Produced in the Liver
- Vitamin K Dependent Factors: Factor II, VII, IX, X, Protein C & S Mn
- Through Gamma Carboxylation of Glutamate Residues
- Half-Life of Vitamin K-Dependent Factors:
- Factor II: 60-72 Hours
- Factor VII: 4-6 Hours (Shortest)
- Factor IX: 21-30 Hours
- Factor X: 48-72 Hours
- Protein C: 6-8 Hours (Second Shortest)
- Protein S: 30-60 Hours
Mediators of Platelet Aggregation
- Von Willebrand Factor (vWF)
- Produced by Endothelium
- Binds to Exposed Collagen at Sites of Vascular Injury for Platelet Adhesion
- Promotes Platelet Aggregation Through GPIb (Most Efficient When Under Shear Stress)
- Thromboxane A2 (TXA2)
- Produced by Activated Platelets
- Increased Platelet Aggregation
- Triggers Calcium Release in Platelets (Exposes GpIIb/IIIa Receptor for Fibrin)
- Induces Vasoconstriction
- Prostacyclin (PGI2/Prostaglandin I2)
- Produced by Endothelium
- Inhibits Platelet Aggregation
- Increases cAMP in Platelets
- Induces Vasodilation
Mediators of Anticoagulation
- Inhibitory Enzymes:
- Antithrombin III (AT-III)
- Inhibits Thrombin (IIa) & Factor Xa
- Activated by Heparin
- Activated Protein C (APC)
- Degrades Factors Va & VIIIa
- Protein S
- Cofactor for Protein C
- Antithrombin III (AT-III)
- Fibrinolysis:
- Tissue Plasminogen Activator (tPA)
- Released from Endothelium
- Converts Plasminogen to Plasmin
- Inhibited by Plasminogen Activator Inhibitor (PAI-1 & PAI-2)
- Plasmin
- Function:
- The Normal Active Clotting Inhibitor (The Most Important Clotting Inhibitor in Plasma)
- Degrades Fibrin (Platelet Plug) into Fibrin Degradation Products
- Also Degrades Factors V, VIII & Fibrinogen
- Plasminogen is Converted to Active Plasmin by tPA, Streptokinase & Urokinase
- Inhibited by α-2 Antiplasmin
- Released from Endothelium
- Decreased Production in Liver Cirrhosis
- Function:
- Tissue Plasminogen Activator (tPA)
Mnemonics
Vitamin K-Dependent Factors
- “2 plus 7 is 9, Knot 10”